Functional and binding data for rat muscarinic cholinergic receptor

• List of ligands
• List of receptors

Ligand	pKi value		Method	Comment
4,5-dihydro-8-methoxy-1H-benz[g]indole -1-ethanamine(E)-2-butenedioate (1:1)	<5.3		1-01201
4-[[[(3-chlorophenyl)amino]carbonyl]oxy]-N,N,N-trimethyl -2-butyn-1-aminiumchloride	5.3		1-01201
GBR 12909 .2HCl	6.2		1-01201
GBR 12909 .2HCl	6.3		1-01202
GBR 12909 .2HCl	6.4		1-01201
KB-2796	5.6		1-01201
amoxapine	6.2		1-01201
aptazapine maleate	6.3		1-01201
benperidol	6.3		1-01201
benzetimide hydrochloride	10.2		1-01201
benzetimide hydrochloride	9.3		1-01201
benzetimide hydrochloride	9.6		1-01201
bupropion HCl	<5.4		1-01202
buspirone HCl	<5.8		1-01201
chlorprothixene HCl H2O	7.8		1-01201
clopenthixol di-HCl (cis)	6.1		1-01201
clopipazan mesylate	7.4		1-01201
clothiapine	6.9		1-01201
cryptopine	4.3		1-01201
dexetimide hydrochloride	11		1-01201
dexetimide hydrochloride	9.8		1-01201
dexetimide hydrochloride	9.9		1-01201
diltiazem hydrochloride	<4.8		1-01201
dixyrazine	5.7		1-01201	REST OF EXPERIMENT IN 83007
dixyrazine	5.8		1-01201	REST OF EXPERIMENT IN 83507
dogmatil	<5		1-01201
droperidol	6.2		1-01201
egyt 3615	4.9		1-01201
fluanisone	5.3		1-01201
flunarizine di-HCl	5.4		1-01201
flupentixol di-HCl (cis)	6.1		1-01201
fluperlapine	7.2		1-01201
ipsapirone	4.6		1-01201
levetimide hydrochloride	5.6		1-01201
levetimide hydrochloride	5.8		1-01201
levetimide hydrochloride	6.1		1-01201
lidoflazine	5.9		1-01201
methotrimeprazine maleate	6.8		1-01201
mianserin HCl (racemate)	6.1		1-01201
mianserin HCl (racemate)	6.2		1-01201
mianserin HCl (racemate)	6.2		1-01201
mianserin HCl (racemate)	6.5		1-01201
mianserin HCl (racemate)	6.5		1-01201
mianserin HCl (racemate)	6.6		1-01201
mianserin HCl R(-)	6.6		1-01201
mianserin HCl R(-)	7		1-01201
mianserin HCl S(+)	5.4		1-01201
mianserin HCl S(+)	5.5		1-01201
mirtazapine HCl (racemate)	5.8		1-01201
mirtazapine HCl (racemate)	5.8		1-01201
mirtazapine HCl (racemate)	6.1		1-01201
mirtazapine HCl (racemate)	6.1		1-01201
mirtazapine HCl (racemate)	6.2		1-01201
mirtazapine HCl (racemate)	6.2		1-01201
mirtazapine HCl (racemate)	6.2		1-01201
mirtazapine HCl (racemate)	6.2		1-01201
mirtazapine HCl R(-)	6.6		1-01201
mirtazapine HCl R(-)	6.7		1-01201
mirtazapine HCl S(+)	5.1		1-01201
mirtazapine HCl S(+)	5.2		1-01201
molindone HCl	<4.8		1-01201
morphine 3-nicotinate HCl	3.9		1-01201
morphine 6-nicotinate HCl	4.7		1-01201
oxiperomide	5.5		1-01201
oxypertine	<6		1-01201
pericyazine	5.9		1-01201
perlapine	7.3		1-01201
pinaverium bromide	6.6		1-01201
pipamperone di-HCl	<6		1-01201
pipotiazine	6.6		1-01201
prothipendyl HCl H2O	6.2		1-01201
risperidone	5.2		1-01201
risperidone	5.5		1-01201
ritanserin	6.1		1-01201
ritanserin	6.1		1-01201
setoperone	5.6		1-01201
spiperone	5.6		1-01201
thioproperazine dimethanesulfonate	6		1-01201
tiapride HCl	<4.9		1-01201
trans-5-chloro-2,3,3a,12b-tetrahydro-2-methyl- 1H-dibenz(2,3:6,7)oxepino(4,5-c)pyrrole maleate	5.3		1-01201
trans-5-chloro-2,3,3a,12b-tetrahydro-2-methyl- 1H-dibenz(2,3:6,7)oxepino(4,5-c)pyrrole maleate	5.3		1-01201
trans-5-chloro-2,3,3a,12b-tetrahydro-2-methyl- 1H-dibenz(2,3:6,7)oxepino(4,5-c)pyrrole maleate	5.3		1-01201
trans-5-chloro-2,3,3a,12b-tetrahydro-2-methyl- 1H-dibenz(2,3:6,7)oxepino(4,5-c)pyrrole maleate	5.8		1-01201
trifluoperazine di-HCl	6.1		1-01201
trifluperidol HCl	4.8		1-01201
triflupromazine HCl	7		1-01201
vilan/nicomorphine HCl	4.7		1-01201