Functional and binding data for rat serotonin 5HT1A receptor

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LigandpKi valueMethodComment
1-(6-chloro-2-pyridinyl)piperazine(E)-2-butenedioate (1:1) salt6.81-02302
1-(6-chloro-2-pyridinyl)piperazine(E)-2-butenedioate (1:1) salt6.81-02302
1-[2-(methylthio)phenyl]piperazine(Z)-2-butenedioate (1:1) salt7.91-02302
1-[2-(methylthio)phenyl]piperazine(Z)-2-butenedioate (1:1) salt8.21-02302


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(C) GPCRDB. F.H., David Lutje Hulsik (D.LutjeHulsik@cmbi.kun.nl), 18-Mar-2002