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| Receptor | Organism | pKi value | pA2 value | pD2 value | Method | Comment | |
|---|---|---|---|---|---|---|---|
| 5HT1A | rat | 7.7 | 1-02301 | ||||
| 5HT1B | rat | 7.8 | 1-02201 | ||||
| 5HT1C | pig | 6.5 | 2-00201 | ||||
| 5HT2B | rat | 6.7 | 1-00502 | MODERATE COMPETITIVE AND NON-COMPETITIVE ANTAGONISM. | |||
| 5HT2B | rat | 6.2 | 1-00502 | MODERATE COMPETITIVE AND NON-COMPETITIVE ANTAGONISM. | |||
| 5HT2B | rat | 8.04 | 1-00502 | MODERATE COMPETITIVE AND NON-COMPETITIVE ANTAGONISM. | |||
| 5HT2C | human | 6.6 | 2-01101 | ||||
| 5HT2C | human | 6.7 | 2-01101 | ||||
| 5HT2C | human | 6.8 | 2-01101 |