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| Receptor | Organism | pKi value | pA2 value | pD2 value | Method | Comment | |
|---|---|---|---|---|---|---|---|
| 5HT1A | human | 8.1 | 2-00601 | ||||
| 5HT1A | human | 8.6 | 2-00601 | ||||
| 5HT1A | human | 8.6 | 2-00601 | ||||
| 5HT1A | rat | 10 | 1-02301 | ||||
| 5HT1A | rat | 8.1 | 1-02301 | ||||
| 5HT1A | rat | >9.1 | 1-02301 | ||||
| 5HT1A | rat | 9.1 | 1-02301 | ||||
| 5HT1B | rat | <5.3 | 1-02201 | ||||
| 5HT2B | rat | 6.06 | 1-00502 | pA2 SCHILD PLOT CALCULATED A MODERATE COMPETITIVE ANTAGONISM | |||
| 5HT2B | rat | 7.93 | 1-00502 | pA2 SCHILD PLOT CALCULATED A MODERATE COMPETITIVE ANTAGONISM | |||
| 5HT2 | rat | 5.4 | 1-02601 | ||||
| AChM | rat | 4.6 | 1-01201 | ||||
| DA | rat | 6.1 | 1-01301 | ||||
| DA | rat | 5.5 | 1-00201 | ||||
| H1 | guinea-pig | 5.8 | 1-00303 | WEAK COMPETITIVE ANTAGONISM. | |||
| H1 | guinea-pig | 6.75 | 1-00303 | WEAK COMPETITIVE ANTAGONISM. | |||
| NAa1 | rat | 7 | 1-02001 | ||||
| NAa1 | rat | 7.76 | 1-01601 | RATHER STRONG COMPETITIVE ANTAGONISM. | |||
| NAa1 | rat | 6.76 | 1-01601 | RATHER STRONG COMPETITIVE ANTAGONISM. | |||
| NAa2 | rat | 6.3 | 1-01501 | ||||
| NAa2 | rat | 6.5 | 1-02101 | MODERATE COMPETITIVE ANTAGONISM AND AT HIGH CONC. A HIGHER T | |||
| NAa2 | rat | 6.05 | 1-02101 | MODERATE COMPETITIVE ANTAGONISM AND AT HIGH CONC. A HIGHER T |