| Receptor | Organism | pKi value | pA2 value | pD2 value | | Method | Comment |
| 5HT2B | rat | | 5.29 | | | 1-00502 | WEAK COMPETITIVE ANTAGONISM AND AT HIGH CONC. A SPASMOGENIC EFFECT. |
| 5HT2B | rat | | | 3.5 | | 1-00502 | VERY VERY WEAK AGONISTIC- AND TACHYPHYLACTIC ACTIVITY. |
| 5HT2B | rat | | | 7.85 | | 1-00502 | WEAK COMPETITIVE ANTAGONISM AND AT HIGH CONC. A SPASMOGENIC EFFECT. |
| 5HT2B | rat | | | 7.8 | | 1-00502 | VERY VERY WEAK AGONISTIC- AND TACHYPHYLACTIC ACTIVITY. |
| 5HT2 | rat | 6.8 | | | | 1-01401 | |
| AChM1 | human | 8.7 | | | | 2-01601 | |
| AChM1 | human | 8.7 | | | | 2-01601 | |
| AChM1 | human | 9 | | | | 2-01601 | |
| AChM2 | human | 7.1 | | | | 2-02001 | |
| AChM2 | human | 7.1 | | | | 2-02001 | |
| AChM2 | human | 7.2 | | | | 2-02001 | |
| AChM | rat | >11 | | | | 1-01901 | |
| AChM | rat | 12.2 | | | | 1-01901 | |
| AChM | rat | >12 | | | | 1-01901 | |
| AChM | rat | >9.1 | | | | 1-01901 | |
| AChM | rat | >9 | | | | 1-01901 | |
| AChM | rat | 7.4 | | | | 1-01801 | |
| AChM | rat | 7.7 | | | | 1-01801 | |
| AChM | rat | 8.2 | | | | 1-01801 | |
| AChM | guinea-pig | | 7.84 | | | 1-01001 | RATHER STRONG COMPETITIVE ANTAGONISM. |
| AChM | guinea-pig | | | 7.27 | | 1-01001 | RATHER STRONG COMPETITIVE ANTAGONISM. |
| DA | rat | 5.6 | | | | 1-01301 | |
| DA | rat | <5.5 | | | | 1-00201 | |
| H1 | guinea-pig | | 5.3 | | | 1-00303 | WEAK COMPETITIVE- AND VERY WEAK NON-COMPETITIVE ANTAGONISM. |
| H1 | guinea-pig | | | 4.5 | | 1-00303 | WEAK COMPETITIVE- AND VERY WEAK NON-COMPETITIVE ANTAGONISM. |
| H1 | guinea-pig | | | 6.56 | | 1-00303 | WEAK COMPETITIVE- AND VERY WEAK NON-COMPETITIVE ANTAGONISM. |
| H2 | guinea-pig | | <5 | | | 1-00902 | NO ANTAGONISTIC ACTIVITY FOUND. AT 1.0E-05 M. A STRONG NEGATIVE CHRONOTROPIC EFFECT. |
| H2 | guinea-pig | | | 5.36 | | 1-00902 | NO ANTAGONISTIC ACTIVITY FOUND. AT 1.0E-05 M. A STRONG NEGATIVE CHRONOTROPIC EFFECT. |
| NAa1 | rat | | | 5.2 | | 1-01601 | WEAK NON-COMPETITIVE ANTAGONISM. |
| NAa1 | rat | | | 6.76 | | 1-01601 | WEAK NON-COMPETITIVE ANTAGONISM. |
| NAa2 | rat | 4.8 | | | | 1-01501 | |
| NAa2 | rat | | 4.5 | | | 1-02101 | VERY WEAK COMPETITIVE ANTAGONISM AND A HIGHER TWITCH-RESPONSE IN HIGH CONCENTRATIONS. |
| NAa2 | rat | | | 6.19 | | 1-02101 | VERY WEAK COMPETITIVE ANTAGONISM AND A HIGHER TWITCH-RESPONSE IN HIGH CONCENTRATIONS. |
| NAa2 | rat | | 5 | | | 1-00601 | pA2 SCHILD PLOT CALCULATED VERY WEAK COMPETITIVE- AND VERY WEAK N0N- COMPETITIVE ANTAGONISM. |
| NAa2 | rat | | | 4.61 | | 1-00601 | pA2 SCHILD PLOT CALCULATED VERY WEAK COMPETITIVE- AND VERY WEAK N0N- COMPETITIVE ANTAGONISM. |
| NAa2 | rat | | | 5.76 | | 1-00601 | pA2 SCHILD PLOT CALCULATED VERY WEAK COMPETITIVE- AND VERY WEAK N0N- COMPETITIVE ANTAGONISM. |
| NAb1 | guinea-pig | | <4.5 | | | 1-00701 | NO ANTAGONISTIC EFFECT FOUND. LETHAL CONC. AT 1E-5M. |
| NAb1 | guinea-pig | | | 7.3 | | 1-00701 | NO ANTAGONISTIC EFFECT FOUND. LETHAL CONC. AT 1E-5M. |
| NAb2 | guinea-pig | | <4.5 | | | 1-00802 | NO ANTAGONISTIC ACTIVITY FOUND AT 3.0E-05 M. |
| NAb2 | guinea-pig | | | 8.2 | | 1-00802 | NO ANTAGONISTIC ACTIVITY FOUND AT 3.0E-05 M. |
Copyright (C) 2002, GPCRDB.