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| Receptor | Organism | pKi value | Method | Comment | |
|---|---|---|---|---|---|
| 5HT1A | rat | >5.6 | 1-02301 | ||
| 5HT1A | rat | 7.2 | 1-02301 | ||
| 5HT1C | pig | >5.8 | 2-00201 | ||
| 5HT1C | pig | 6.6 | 2-00201 | ||
| 5HT2 | rat | <5.8 | 1-02601 | ||
| 5HT2C | human | 5.9 | 2-01101 | ||
| 5HT2C | human | 5.9 | 2-01101 | ||
| 5HT2C | human | 6.1 | 2-01101 | ||
| AChM | rat | <5.8 | 1-02501 | ||
| DA1 | rat | <5.7 | 1-02401 | ||
| DA | rat | <5.9 | 1-00201 | ||
| NAa2 | rat | >5.6 | 1-01501 | ||
| NAa2 | rat | 6.2 | 1-01501 | ||
| NAa2 | rat | 6.5 | 1-01501 |