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| Receptor | Organism | pKi value | pA2 value | pD2 value | Method | Comment | |
|---|---|---|---|---|---|---|---|
| 5HT2B | rat | 6.9 | 1-00502 | pA2 SCHILD-PLOT CALCULATED RATHER STRONG COMPETITIVE ANTAGONISM. | |||
| 5HT2B | rat | 7.88 | 1-00502 | pA2 SCHILD-PLOT CALCULATED RATHER STRONG COMPETITIVE ANTAGONISM. | |||
| 5HT2 | rat | 7 | 1-01401 | ||||
| AChM | rat | 6.1 | 1-01201 | ||||
| DA | rat | 8.4 | 1-00201 | ||||
| DA | rat | 9.6 | 1-00201 | ||||
| H1 | rat | 8.1 | 1-01101 | ||||
| H1 | rat | 8 | 1-01101 | ||||
| NAa2 | rat | 7.6 | 1-00601 | SHOWED A RATHER STRONG COMPETITIVE ANTAGONISM TO NA ON ALPHA-ADRENERGIC RECEPTORS. | |||
| NAa2 | rat | 5.3 | 1-00601 | SHOWED A RATHER STRONG COMPETITIVE ANTAGONISM TO NA ON ALPHA-ADRENERGIC RECEPTORS. | |||
| NAa | rat | 7.1 | 1-00101 |