Functional and binding data for olanzapine
Copyright (C) 2002,
GPCRDB
.
List of
ligands
List of
receptors
Receptor
Organism
pK
i
value
pA
2
value
pD
2
value
Method
Comment
5HT1A
human
5.6
2-01801
5HT1A
human
5.9
2-01801
5HT1A
human
6
2-01801
5HT1A
human
6
2-01801
5HT2A
human
7.8
2-01901
5HT2A
human
7.8
2-01901
5HT2A
human
7.9
2-01901
5HT2A
human
8.1
2-01901
5HT2A
human
8.6
2-01901
5HT2A
human
8.7
2-01901
5HT2A
human
8.8
2-01901
5HT2A
human
8.8
2-01901
5HT2A
human
8.9
2-01901
5HT2A
human
8.9
2-01901
5HT2A
human
8.9
2-01201
5HT2A
human
>8
2-01201
5HT2B
rat
7.2
1-00502
5HT2B
rat
8.1
1-00502
5HT2C
human
7.8
2-01101
5HT2C
human
8.1
2-01101
AChM1
human
7.1
2-01601
AChM1
human
7.5
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.7
2-01601
AChM1
human
7.8
2-01601
AChM1
human
7.8
2-01601
AChM1
human
7.9
2-01601
AChM1
human
8.3
2-01601
AChM2
human
6.7
2-02001
AChM2
human
6.7
2-02001
AChM2
human
6.7
2-02001
AChM2
human
6.7
2-02001
AChM2
human
6.8
2-02001
AChM2
human
7
2-02001
AChM2
guinea-pig
6.7
2-00101
AChM2
guinea-pig
6.8
2-00101
AChM
rat
7.8
1-01203
AChM
rat
8.1
1-01203
AChM
rat
8.2
1-01203
AChM
rat
8
1-01203
AChM
rat
8
1-01203
AChM
rat
8
1-01203
AChM
rat
8
1-01203
AChM
rat
8
1-01203
AChM
guinea-pig
6.8
1-01001
AChM
guinea-pig
7
1-01001
DA1
rat
7.2
1-02403
DA1
rat
7.2
1-02403
DA1
rat
7.2
1-02403
DA1
rat
7.3
1-02403
DA1
rat
7.4
1-02403
DA1
rat
7.6
1-02403
DA1
rat
7.6
1-02403
DA1
rat
7.7
1-02403
DA1
rat
7.8
1-02403
DA1
rat
8.4
1-02403
DA1
rat
8.5
1-02403
DA2B
human
6.9
2-01701
DA2B
human
7.1
2-01701
DA2B
human
7.3
2-01701
DA2B
human
7.4
2-01701
DA2B
human
7.5
2-01701
DA2B
human
7.5
2-01701
DA2B
human
7.7
2-01701
DA2B
human
7.7
2-01701
DA2B
human
7.8
2-01701
DA2B
human
7.8
2-01701
DA2B
human
7.9
2-01701
DA2B
human
7.9
2-01701
DA2B
human
7.9
2-01701
DA2B
human
7.9
2-01701
DA2B
human
7
2-01701
DA2
rat
7.2
1-00203
DA2
rat
7.2
1-00203
DA2
rat
7.5
1-00203
DA2
rat
7.5
1-00203
DA2
rat
7.7
1-00203
DA2
rat
8.4
1-00203
low hill slope
DA2
rat
>8
1-00203
LOW HILL SLOPE
DA2
rat
9.3
1-00203
H1
guinea-pig
8.5
2-02101
H1
guinea-pig
8.6
2-02101
H1
guinea-pig
8.6
2-02101
H1
guinea-pig
8.6
2-02101
H1
guinea-pig
8.7
2-02101
H1
guinea-pig
8.8
2-02101
NAa1
rat
6.3
2-02201
NAa1
rat
6.3
2-02201
NAa1
rat
6.4
2-02201
NAa1
rat
6.5
2-02201
NAa1
rat
6.6
2-02201
NAa1
rat
6.7
2-02201
NAa1
rat
6.7
2-02201
NAa1
rat
6.8
2-02201
NAa1
rat
6.9
2-02201
NAa1
rat
7.3
2-02201
NAa1
rat
7
2-02201
NAa1
rat
7.6
1-02001
(C) GPCRDB. F.H., David Lutje Hulsik (D.LutjeHulsik@cmbi.kun.nl), 18-Mar-2002