Functional and binding data for olanzapine

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ReceptorOrganismpKi valuepA2 valuepD2 valueMethodComment
5HT1Ahuman5.62-01801
5HT1Ahuman5.92-01801
5HT1Ahuman62-01801
5HT1Ahuman62-01801
5HT2Ahuman7.82-01901
5HT2Ahuman7.82-01901
5HT2Ahuman7.92-01901
5HT2Ahuman8.12-01901
5HT2Ahuman8.62-01901
5HT2Ahuman8.72-01901
5HT2Ahuman8.82-01901
5HT2Ahuman8.82-01901
5HT2Ahuman8.92-01901
5HT2Ahuman8.92-01901
5HT2Ahuman8.92-01201
5HT2Ahuman>82-01201
5HT2Brat7.21-00502
5HT2Brat8.11-00502
5HT2Chuman7.82-01101
5HT2Chuman8.12-01101
AChM1human7.12-01601
AChM1human7.52-01601
AChM1human7.72-01601
AChM1human7.72-01601
AChM1human7.72-01601
AChM1human7.72-01601
AChM1human7.72-01601
AChM1human7.72-01601
AChM1human7.82-01601
AChM1human7.82-01601
AChM1human7.92-01601
AChM1human8.32-01601
AChM2human6.72-02001
AChM2human6.72-02001
AChM2human6.72-02001
AChM2human6.72-02001
AChM2human6.82-02001
AChM2human72-02001
AChM2guinea-pig6.72-00101
AChM2guinea-pig6.82-00101
AChMrat7.81-01203
AChMrat8.11-01203
AChMrat8.21-01203
AChMrat81-01203
AChMrat81-01203
AChMrat81-01203
AChMrat81-01203
AChMrat81-01203
AChMguinea-pig6.81-01001
AChMguinea-pig71-01001
DA1rat7.21-02403
DA1rat7.21-02403
DA1rat7.21-02403
DA1rat7.31-02403
DA1rat7.41-02403
DA1rat7.61-02403
DA1rat7.61-02403
DA1rat7.71-02403
DA1rat7.81-02403
DA1rat8.41-02403
DA1rat8.51-02403
DA2Bhuman6.92-01701
DA2Bhuman7.12-01701
DA2Bhuman7.32-01701
DA2Bhuman7.42-01701
DA2Bhuman7.52-01701
DA2Bhuman7.52-01701
DA2Bhuman7.72-01701
DA2Bhuman7.72-01701
DA2Bhuman7.82-01701
DA2Bhuman7.82-01701
DA2Bhuman7.92-01701
DA2Bhuman7.92-01701
DA2Bhuman7.92-01701
DA2Bhuman7.92-01701
DA2Bhuman72-01701
DA2rat7.21-00203
DA2rat7.21-00203
DA2rat7.51-00203
DA2rat7.51-00203
DA2rat7.71-00203
DA2rat8.41-00203low hill slope
DA2rat>81-00203LOW HILL SLOPE
DA2rat9.31-00203
H1guinea-pig8.52-02101
H1guinea-pig8.62-02101
H1guinea-pig8.62-02101
H1guinea-pig8.62-02101
H1guinea-pig8.72-02101
H1guinea-pig8.82-02101
NAa1rat6.32-02201
NAa1rat6.32-02201
NAa1rat6.42-02201
NAa1rat6.52-02201
NAa1rat6.62-02201
NAa1rat6.72-02201
NAa1rat6.72-02201
NAa1rat6.82-02201
NAa1rat6.92-02201
NAa1rat7.32-02201
NAa1rat72-02201
NAa1rat7.61-02001


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(C) GPCRDB. F.H., David Lutje Hulsik (D.LutjeHulsik@cmbi.kun.nl), 18-Mar-2002